In vitro antibacterial activities of silver (I) 4-substituted benzenesulfonate derivatives

A new series of silver (I) 4-substitutedbenzenesulfonate derivatives (1-8) have been synthesized in order to search for new potential antibacterial agents. The antibacterial activity of 1-8 against various strains of bacteria has been determined. Compounds 2-4 (silver (I) 4-methylbenzenesulfonate...

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Autores principales: Chanawanno, Kullapa, Chantrapromma, Suchada, Anantapong, Theerasak, Kanjana-Opas, Akkharawit
Formato: Articulo
Lenguaje:Inglés
Publicado: 2010
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Acceso en línea:http://sedici.unlp.edu.ar/handle/10915/8044
http://www.latamjpharm.org/resumenes/29/7/LAJOP_29_7_1_17.pdf
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Sumario:A new series of silver (I) 4-substitutedbenzenesulfonate derivatives (1-8) have been synthesized in order to search for new potential antibacterial agents. The antibacterial activity of 1-8 against various strains of bacteria has been determined. Compounds 2-4 (silver (I) 4-methylbenzenesulfonate (2), silver (I) 4-methoxybenzenesulfonate (3), and silver (I) 4-aminobenzenesulfonate (4)) showed broad spectrum of antibacterial activities against both Gram-positive (methicillin-resistant Staphylococcus aureus, Staphylococcus aureus, Bacillus subtilis, Enterococcus faecalis and vancomycin-resistant Enterococcus faecalis) and only one Gram-negative bacterium (Shigella sonnei). The Structure-Activity Relationship (SAR) has also been reported.